PDB 5usq
PDB Information
| PDB | 5USQ |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Design, synthesis and optimization of 7-substituted-pyrazolo[4,3-b]pyridine ALK5 (activin receptor-like kinase 5) inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-02-13 |
| Resolution | 2.550 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5usqA01 | 25 May, 2017 | 3.30.200.20 | Assigned |
| 5usqA02 | 25 May, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P36897 | TGFR1_HUMAN | Homo sapiens | TGF-beta receptor type-1 |
