PDB 5ur1
PDB Information
| PDB | 5UR1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | 2-Oxo-3, 4-dihydropyrimido[4, 5-d]pyrimidinyl derivatives as new irreversible pan fibroblast growth factor receptor (FGFR) inhibitors.
Eur J Med Chem
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-02-09 |
| Resolution | 2.200 |
| CATH Insert Date | 14 Nov, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Nov, 2017 | Chopped |
| B | 14 Nov, 2017 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5ur1A01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5ur1A02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
| 5ur1B01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5ur1B02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |
| P11362 | FGFR1_HUMAN | Homo sapiens | Fibroblast growth factor receptor 1 |
