PDB Information

PDB5UOY
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Selective Phosphodiesterase 1 Inhibitors with Memory Enhancing Properties.
Dyck, B., Branstetter, B., Gharbaoui, T., Hudson, A.R., Breitenbucher, J.G., Gomez, L., Botrous, I., Marrone, T., Barido, R., Allerston, C.K., Cedervall, E.P., Xu, R., Sridhar, V., Barker, R., Aertgeerts, K., Schmelzer, K., Neul, D., Lee, D., Massari, M.E., Andersen, C.B., Sebring, K., Zhou, X., Petroski, R., Limberis, J., Augustin, M., Chun, L.E., Edwards, T.E., Peters, M., Tabatabaei, A.
J. Med. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-02-01
Resolution1.820
CATH Insert Date07 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5uoyA00 25 May, 2017 1.10.1300.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q01064 PDE1B_HUMAN Homo sapiens Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B