PDB 5uob
PDB Information
| PDB | 5UOB |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Nitrile in the Hole: Discovery of a Small Auxiliary Pocket in Neuronal Nitric Oxide Synthase Leading to the Development of Potent and Selective 2-Aminoquinoline Inhibitors.
J. Med. Chem.
|
| Header | Oxidoreductase/Oxidoreductase Inhibitor |
| Released | 2017-01-31 |
| Resolution | 2.290 |
| CATH Insert Date | 14 May, 2017 |
PDB Images (17)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 May, 2017 | Chopped |
| B | 15 May, 2017 | Chopped |
| C | 15 May, 2017 | Chopped |
| D | 15 May, 2017 | Chopped |
CATH Domains (12)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5uobA01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uobA02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uobA03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uobB01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uobB02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uobB03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uobC01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uobC02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uobC03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uobD01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uobD02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uobD03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
