PDB 5uo9
PDB Information
| PDB | 5UO9 |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | Homo sapiens |
| Primary Citation | Nitrile in the Hole: Discovery of a Small Auxiliary Pocket in Neuronal Nitric Oxide Synthase Leading to the Development of Potent and Selective 2-Aminoquinoline Inhibitors.
J. Med. Chem.
|
| Header | Oxidoreductase/Oxidoreductase Inhibitor |
| Released | 2017-01-31 |
| Resolution | 2.190 |
| CATH Insert Date | 14 May, 2017 |
PDB Images (17)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 May, 2017 | Chopped |
| B | 15 May, 2017 | Chopped |
| C | 15 May, 2017 | Chopped |
| D | 15 May, 2017 | Chopped |
CATH Domains (12)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5uo9A01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uo9A02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uo9A03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uo9B01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uo9B02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uo9B03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uo9C01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uo9C02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uo9C03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
| 5uo9D01 | 06 Nov, 2017 | 3.90.340.10 | Assigned |
| 5uo9D02 | 06 Nov, 2017 | 3.90.440.10 | Assigned |
| 5uo9D03 | 06 Nov, 2017 | 3.90.1230.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
| P29474 | NOS3_HUMAN | Homo sapiens | Nitric oxide synthase, endothelial |
