PDB 5u7q
PDB Information
| PDB | 5U7Q |
| Method | X-RAY DIFFRACTION |
| Host Organism | Baculovirus expression vector pFastBac1-HM |
| Gene Source | Homo sapiens |
| Primary Citation | Identification of a new class of potent Cdc7 inhibitors designed by putative pharmacophore model: Synthesis and biological evaluation of 2,3-dihydrothieno[3,2-d]pyrimidin-4(1H)-ones.
Bioorg. Med. Chem.
|
| Header | Transferase |
| Released | 2016-12-12 |
| Resolution | 3.150 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
| C | 08 May, 2017 | Chopped |
| D | 08 May, 2017 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5u7qA01 | 07 Mar, 2018 | 3.30.200.20 | Assigned |
| 5u7qA02 | 07 Mar, 2018 | 1.10.510.10 | Assigned |
| 5u7qB01 | 07 Mar, 2018 | 3.30.200.20 | Assigned |
| 5u7qB02 | 07 Mar, 2018 | 1.10.510.10 | Assigned |
| 5u7qC01 | 07 Mar, 2018 | 3.30.200.20 | Assigned |
| 5u7qC02 | 07 Mar, 2018 | 1.10.510.10 | Assigned |
| 5u7qD01 | 07 Mar, 2018 | 3.30.200.20 | Assigned |
| 5u7qD02 | 07 Mar, 2018 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O75116 | ROCK2_HUMAN | Homo sapiens | Rho-associated protein kinase 2 |
| O75116 | ROCK2_HUMAN | Homo sapiens | Rho-associated protein kinase 2 |
| O75116 | ROCK2_HUMAN | Homo sapiens | Rho-associated protein kinase 2 |
| O75116 | ROCK2_HUMAN | Homo sapiens | Rho-associated protein kinase 2 |
