PDB 5u2c

PDB Links
Overview

PDB Information

PDB	5U2C
Method	X-RAY DIFFRACTION
Host Organism	Escherichia coli
Gene Source	Homo sapiens
Primary Citation	Dual-activity PI3K-BRD4 inhibitor for the orthogonal inhibition of MYC to block tumor growth and metastasis. Andrews, F.H., Singh, A.R., Joshi, S., Smith, C.A., Morales, G.A., Garlich, J.R., Durden, D.L., Kutateladze, T.G. Proc. Natl. Acad. Sci. U.S.A.
Header	Transcription Regulator/Inhibitor
Released	2016-11-30
Resolution	3.300
CATH Insert Date	07 May, 2017

PDB Images (5)

Image of CATH 5u2c

5u2c

PDB 5u2c

Image of CATH 5u2cA

5u2cA

PDB Chain 5u2cA

Image of CATH 5u2cB

5u2cB

PDB Chain 5u2cB

Image of CATH 5u2cA00

5u2cA00

CATH Domain 5u2cA00

Image of CATH 5u2cB00

5u2cB00

CATH Domain 5u2cB00

PDB Prints

PDB Chains (2)

Chain ID	Date inserted into CATH	CATH Status
A	08 May, 2017	Chopped
B	08 May, 2017	Chopped

CATH Domains (2)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
5u2cA00	23 May, 2017	1.20.920.10	Assigned
5u2cB00	23 May, 2017	1.20.920.10	Assigned

UniProtKB Entries (2)

Accession	Gene ID	Taxon	Description
O60885	BRD4_HUMAN	Homo sapiens	Bromodomain-containing protein 4
O60885	BRD4_HUMAN	Homo sapiens	Bromodomain-containing protein 4