PDB 5u1q
PDB Information
| PDB | 5U1Q |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target.
J. Med. Chem.
|
| Header | Signaling Protein/Peptide Inhibitor |
| Released | 2016-11-28 |
| Resolution | 2.100 |
| CATH Insert Date | 17 Dec, 2017 |
PDB Images (13)
PDB Prints
PDB Chains (8)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 17 Dec, 2017 | Chopped |
| B | 17 Dec, 2017 | Chopped |
| C | 17 Dec, 2017 | Chopped |
| D | 17 Dec, 2017 | Chopped |
| L | 17 Dec, 2017 | Rejected |
| M | 17 Dec, 2017 | Rejected |
| N | 17 Dec, 2017 | Rejected |
| P | 17 Dec, 2017 | Rejected |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5u1qA00 | 22 Dec, 2017 | 3.30.505.10 | Assigned |
| 5u1qB00 | 22 Dec, 2017 | 3.30.505.10 | Assigned |
| 5u1qC00 | 22 Dec, 2017 | 3.30.505.10 | Assigned |
| 5u1qD00 | 22 Dec, 2017 | 3.30.505.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q14451 | GRB7_HUMAN | Homo sapiens | Growth factor receptor-bound protein 7 |
| Q14451 | GRB7_HUMAN | Homo sapiens | Growth factor receptor-bound protein 7 |
| Q14451 | GRB7_HUMAN | Homo sapiens | Growth factor receptor-bound protein 7 |
| Q14451 | GRB7_HUMAN | Homo sapiens | Growth factor receptor-bound protein 7 |
