PDB 5th7
PDB Information
| PDB | 5TH7 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase.
J. Med. Chem.
|
| Header | Transferase |
| Released | 2016-09-29 |
| Resolution | 1.950 |
| CATH Insert Date | 20 Nov, 2016 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 21 Nov, 2016 | Chopped |
| B | 21 Nov, 2016 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5th7A00 | 16 Feb, 2017 | 2.170.270.10 | Assigned |
| 5th7B00 | 16 Feb, 2017 | 2.170.270.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9NQR1 | KMT5A_HUMAN | Homo sapiens | N-lysine methyltransferase KMT5A |
| Q9NQR1 | KMT5A_HUMAN | Homo sapiens | N-lysine methyltransferase KMT5A |
