PDB Information

PDB5TF9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K-12
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of Allosteric WNK Kinase Inhibitors.
Yamada, K., Zhang, J.H., Xie, X., Reinhardt, J., Xie, A.Q., LaSala, D., Kohls, D., Yowe, D., Burdick, D., Yoshisue, H., Wakai, H., Schmidt, I., Gunawan, J., Yasoshima, K., Yue, Q.K., Kato, M., Mogi, M., Idamakanti, N., Kreder, N., Drueckes, P., Pandey, P., Kawanami, T., Huang, W., Yagi, Y.I., Deng, Z., Park, H.M.
ACS Chem. Biol.
HeaderTransferase/Transferase Inhibitor
Released2016-09-24
Resolution2.500
CATH Insert Date06 Nov, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Nov, 2016 Chopped
B 07 Nov, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5tf9A01 10 Nov, 2016 3.30.200.20 Assigned
5tf9A02 10 Nov, 2016 1.10.510.10 Assigned
5tf9B01 10 Nov, 2016 3.30.200.20 Assigned
5tf9B02 10 Nov, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H4A3 WNK1_HUMAN Homo sapiens Serine/threonine-protein kinase WNK1
Q9H4A3 WNK1_HUMAN Homo sapiens Serine/threonine-protein kinase WNK1