PDB 5td2
PDB Information
| PDB | 5TD2 | 
| Method | X-RAY DIFFRACTION | 
| Host Organism | Escherichia coli | 
| Gene Source | Homo sapiens | 
| Primary Citation | Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogate. Bioorg. Med. Chem. Lett. | 
| Header | Transferase/Transferase Inhibitor | 
| Released | 2016-09-16 | 
| Resolution | 2.680 | 
| CATH Insert Date | 07 May, 2017 | 
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status | 
|---|---|---|
| A | 08 May, 2017 | Chopped | 
| B | 08 May, 2017 | Chopped | 
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status | 
|---|---|---|---|
| 5td2A01 | 21 May, 2017 | Holding pen | |
| 5td2A02 | 21 May, 2017 | 1.10.510.10 | Assigned | 
| 5td2B01 | 21 May, 2017 | Holding pen | |
| 5td2B02 | 21 May, 2017 | 1.10.510.10 | Assigned | 
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description | 
|---|---|---|---|
| Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer | 
| Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer | 
