PDB Information

PDB5T7F
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
The Discovery of GS-9901: A Potent, Selective and Metabolically Stable Inhibitor of PI3Kd
Patel, L., Chandrasekhar, J., Evarts, J., Forseth, K., Haran, A., Ip, C., Kashishian, A., Kim, M., Koditek, D., Koppenol, S., Lad, L., Lepist, E.-I., McGrath, M.E., Perreault, S., Puri, K., Villasenor, A., Somoza, J.R., Steiner, B., Therrien, J., Trilberg, J., Phillips, G.
To Be Published
HeaderTransferase/Transferase Inhibitor
Released2016-09-04
Resolution2.600
CATH Insert Date08 Jan, 2017

PDB Images (8)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2017 Holding pen
B 09 Jan, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5t7fB01 20 Jan, 2017 1.25.40.70 Assigned
5t7fB02 20 Jan, 2017 3.10.20.90 Assigned
5t7fB03 20 Jan, 2017 2.60.40.150 Assigned
5t7fB04 20 Jan, 2017 3.30.1010.10 Assigned
5t7fB05 20 Jan, 2017 1.10.1070.11 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
CATH-Gene3D is a Global Biodata Core Resource Learn more...