PDB Information

PDB5T5G
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase.
Butler, K.V., Ma, A., Yu, W., Li, F., Tempel, W., Babault, N., Pittella-Silva, F., Shao, J., Wang, J., Luo, M., Vedadi, M., Brown, P.J., Arrowsmith, C.H., Jin, J.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2016-08-30
Resolution2.100
CATH Insert Date09 Oct, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5t5gA00 16 Feb, 2017 2.170.270.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9NQR1 KMT5A_HUMAN Homo sapiens N-lysine methyltransferase KMT5A