PDB 5t5g
PDB Information
| PDB | 5T5G |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase.
J. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2016-08-30 |
| Resolution | 2.100 |
| CATH Insert Date | 09 Oct, 2016 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 10 Oct, 2016 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5t5gA00 | 16 Feb, 2017 | 2.170.270.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9NQR1 | KMT5A_HUMAN | Homo sapiens | N-lysine methyltransferase KMT5A |
