PDB Information

PDB5QJ2
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Potent Triazolopyridine Myeloperoxidase Inhibitors.
Wurtz, N.R., Viet, A., Shaw, S.A., Dilger, A., Valente, M.N., Khan, J.A., Jusuf, S., Narayanan, R., Fernando, G., Lo, F., Liu, X., Locke, G.A., Kopcho, L., Abell, L.M., Sleph, P., Basso, M., Zhao, L., Wexler, R.R., Duclos, F., Kick, E.K.
ACS Med Chem Lett
HeaderMetal Binding Protein
Released2018-09-26
Resolution2.820
CATH Insert Date10 Feb, 2019

PDB Images (17)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 10 Feb, 2019 Chopped
B 10 Feb, 2019 Chopped
D 10 Feb, 2019 Chopped
E 10 Feb, 2019 Chopped
F 10 Feb, 2019 Chopped
G 10 Feb, 2019 Chopped
H 10 Feb, 2019 Chopped
I 10 Feb, 2019 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5qj2A00 11 Feb, 2019 Holding pen
5qj2B00 11 Feb, 2019 1.10.640.10 Assigned
5qj2D00 11 Feb, 2019 Holding pen
5qj2E00 11 Feb, 2019 1.10.640.10 Assigned
5qj2F00 11 Feb, 2019 Holding pen
5qj2G00 11 Feb, 2019 1.10.640.10 Assigned
5qj2H00 11 Feb, 2019 Holding pen
5qj2I00 11 Feb, 2019 1.10.640.10 Assigned

UniProtKB Entries (8)

Accession Gene ID Taxon Description
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase
P05164 PERM_HUMAN Homo sapiens Myeloperoxidase