PDB Information

PDB5OKT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery of Inhibitor of Wnt Production 2 (IWP-2) and Related Compounds As Selective ATP-Competitive Inhibitors of Casein Kinase 1 (CK1) delta / epsilon.
Garcia-Reyes, B., Witt, L., Jansen, B., Karasu, E., Gehring, T., Leban, J., Henne-Bruns, D., Pichlo, C., Brunstein, E., Baumann, U., Wesseler, F., Rathmer, B., Schade, D., Peifer, C., Knippschild, U.
J. Med. Chem.
HeaderTransferase
Released2017-07-25
Resolution2.130
CATH Insert Date03 Jun, 2018

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped
C 03 Jun, 2018 Chopped
D 03 Jun, 2018 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5oktA01 27 Jun, 2018 3.30.200.20 Assigned
5oktA02 27 Jun, 2018 1.10.510.10 Assigned
5oktB01 27 Jun, 2018 3.30.200.20 Assigned
5oktB02 27 Jun, 2018 1.10.510.10 Assigned
5oktC01 27 Jun, 2018 3.30.200.20 Assigned
5oktC02 27 Jun, 2018 1.10.510.10 Assigned
5oktD01 27 Jun, 2018 3.30.200.20 Assigned
5oktD02 27 Jun, 2018 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta