PDB Information

PDB5O83
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Discovery of CDZ173 (Leniolisib), Representing a Structurally Novel Class of PI3K Delta-Selective Inhibitors.
Hoegenauer, K., Soldermann, N., Zecri, F., Strang, R.S., Graveleau, N., Wolf, R.M., Cooke, N.G., Smith, A.B., Hollingworth, G.J., Blanz, J., Gutmann, S., Rummel, G., Littlewood-Evans, A., Burkhart, C.
ACS Med Chem Lett
HeaderTransferase
Released2017-06-12
Resolution2.900
CATH Insert Date14 Nov, 2017

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform