PDB 5nxe
PDB Information
| PDB | 5NXE |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | 2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors.
Sci Rep
|
| Header | Transferase |
| Released | 2017-05-10 |
| Resolution | 1.600 |
| CATH Insert Date | 03 Jun, 2018 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Jun, 2018 | Chopped |
| B | 03 Jun, 2018 | Chopped |
| H | 03 Jun, 2018 | Chopped |
| I | 03 Jun, 2018 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5nxeA00 | 27 Jun, 2018 | 3.90.228.10 | Assigned |
| 5nxeB00 | 27 Jun, 2018 | 3.90.228.10 | Assigned |
| 5nxeH00 | 27 Jun, 2018 | 6.20.320.10 | Assigned |
| 5nxeI00 | 27 Jun, 2018 | 6.20.320.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
