PDB Information

PDB5NCZ
MethodX-RAY DIFFRACTION
Host OrganismInsect cell expression vector pTIE1
Gene SourceMus musculus
Primary Citation
Design and Synthesis of Soluble and Cell-Permeable PI3K delta Inhibitors for Long-Acting Inhaled Administration.
Perry, M.W.D., Bjorhall, K., Bonn, B., Carlsson, J., Chen, Y., Eriksson, A., Fredlund, L., Hao, H., Holden, N.S., Karabelas, K., Lindmark, H., Liu, F., Pemberton, N., Petersen, J., Rodrigo Blomqvist, S., Smith, R.W., Svensson, T., Terstiege, I., Tyrchan, C., Yang, W., Zhao, S., Oster, L.
J. Med. Chem.
HeaderTransferase
Released2017-03-06
Resolution1.940
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5nczA01 10 Dec, 2017 1.25.40.70 Assigned
5nczA02 10 Dec, 2017 3.10.20.90 Assigned
5nczA03 10 Dec, 2017 2.60.40.150 Assigned
5nczA04 10 Dec, 2017 3.30.1010.10 Assigned
5nczA05 10 Dec, 2017 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform