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PDB Information

PDB5MWP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Preclinical pharmacology of AZD9977: A novel mineralocorticoid receptor modulator separating organ protection from effects on electrolyte excretion.
Bamberg, K., Johansson, U., Edman, K., William-Olsson, L., Myhre, S., Gunnarsson, A., Geschwindner, S., Aagaard, A., Bjornson Granqvist, A., Jaisser, F., Huang, Y., Granberg, K.L., Jansson-Lofmark, R., Hartleib-Geschwindner, J.
PLoS ONE
HeaderSignaling Protein
Released2017-01-19
Resolution1.820
CATH Insert Date03 Jun, 2018

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5mwpA00 27 Jun, 2018 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
P08235 MCR_HUMAN Homo sapiens Mineralocorticoid receptor
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