PDB 5mqv
PDB Information
PDB | 5MQV |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21(DE3) |
Gene Source | Homo sapiens |
Primary Citation | Optimized 4,5-Diarylimidazoles as Potent/Selective Inhibitors of Protein Kinase CK1 delta and Their Structural Relation to p38 alpha MAPK.
Molecules
|
Header | Transferase |
Released | 2016-12-20 |
Resolution | 2.150 |
CATH Insert Date | 07 May, 2017 |
PDB Images (19)
PDB Prints
PDB Chains (6)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 May, 2017 | Chopped |
B | 08 May, 2017 | Chopped |
C | 08 May, 2017 | Chopped |
D | 08 May, 2017 | Chopped |
E | 08 May, 2017 | Chopped |
F | 08 May, 2017 | Chopped |
CATH Domains (12)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5mqvA01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvA02 | 17 May, 2017 | 1.10.510.10 | Assigned |
5mqvB01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvB02 | 17 May, 2017 | 1.10.510.10 | Assigned |
5mqvC01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvC02 | 17 May, 2017 | 1.10.510.10 | Assigned |
5mqvD01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvD02 | 17 May, 2017 | 1.10.510.10 | Assigned |
5mqvE01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvE02 | 17 May, 2017 | 1.10.510.10 | Assigned |
5mqvF01 | 17 May, 2017 | 3.30.200.20 | Assigned |
5mqvF02 | 17 May, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (6)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |