PDB Information

PDB5MQV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Optimized 4,5-Diarylimidazoles as Potent/Selective Inhibitors of Protein Kinase CK1 delta and Their Structural Relation to p38 alpha MAPK.
Halekotte, J., Witt, L., Ianes, C., Kruger, M., Buhrmann, M., Rauh, D., Pichlo, C., Brunstein, E., Luxenburger, A., Baumann, U., Knippschild, U., Bischof, J., Peifer, C.
Molecules
HeaderTransferase
Released2016-12-20
Resolution2.150
CATH Insert Date07 May, 2017

PDB Images (19)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
C 08 May, 2017 Chopped
D 08 May, 2017 Chopped
E 08 May, 2017 Chopped
F 08 May, 2017 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
5mqvA01 17 May, 2017 3.30.200.20 Assigned
5mqvA02 17 May, 2017 1.10.510.10 Assigned
5mqvB01 17 May, 2017 3.30.200.20 Assigned
5mqvB02 17 May, 2017 1.10.510.10 Assigned
5mqvC01 17 May, 2017 3.30.200.20 Assigned
5mqvC02 17 May, 2017 1.10.510.10 Assigned
5mqvD01 17 May, 2017 3.30.200.20 Assigned
5mqvD02 17 May, 2017 1.10.510.10 Assigned
5mqvE01 17 May, 2017 3.30.200.20 Assigned
5mqvE02 17 May, 2017 1.10.510.10 Assigned
5mqvF01 17 May, 2017 3.30.200.20 Assigned
5mqvF02 17 May, 2017 1.10.510.10 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta