PDB Information

PDB5MHQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Molecular profiling and combinatorial activity of CCT068127: a potent CDK2 and CDK9 inhibitor.
Whittaker, S.R., Barlow, C., Martin, M.P., Mancusi, C., Wagner, S., Self, A., Barrie, E., Te Poele, R., Sharp, S., Brown, N., Wilson, S., Jackson, W., Fischer, P.M., Clarke, P.A., Walton, M.I., McDonald, E., Blagg, J., Noble, M., Garrett, M.D., Workman, P.
Mol Oncol
HeaderCell Cycle/Inhibitor
Released2016-11-25
Resolution1.300
CATH Insert Date07 Jan, 2018

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jan, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5mhqA01 11 Jan, 2018 3.30.200.20 Assigned
5mhqA02 11 Jan, 2018 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2