PDB Information

PDB5M6U
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of a Potent, Selective, and Orally Available PI3K delta Inhibitor for the Treatment of Inflammatory Diseases.
Erra, M., Taltavull, J., Greco, A., Bernal, F.J., Caturla, J.F., Gracia, J., Dominguez, M., Sabate, M., Paris, S., Soria, S., Hernandez, B., Armengol, C., Cabedo, J., Bravo, M., Calama, E., Miralpeix, M., Lehner, M.D.
ACS Med Chem Lett
HeaderTransferase
Released2016-10-26
Resolution2.850
CATH Insert Date07 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Holding pen
B 08 May, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P27986 P85A_HUMAN Homo sapiens Phosphatidylinositol 3-kinase regulatory subunit alpha
O00329 PK3CD_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform