PDB 5m2v
PDB Information
| PDB | 5M2V |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Rattus norvegicus |
| Primary Citation | Design and Synthesis of a Series of l-trans-4-Substituted Prolines as Selective Antagonists for the Ionotropic Glutamate Receptors Including Functional and X-ray Crystallographic Studies of New Subtype Selective Kainic Acid Receptor Subtype 1 (GluK1) Antagonist (2S,4R)-4-(2-Carboxyphenoxy)pyrrolidine-2-carboxylic Acid.
J. Med. Chem.
|
| Header | Membrane Protein |
| Released | 2016-10-13 |
| Resolution | 3.180 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5m2vA01 | 15 May, 2017 | 3.40.190.10 | Assigned |
| 5m2vA02 | 15 May, 2017 | 3.40.190.10 | Assigned |
| 5m2vB01 | 15 May, 2017 | 3.40.190.10 | Assigned |
| 5m2vB02 | 15 May, 2017 | 3.40.190.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P22756 | GRIK1_RAT | Rattus norvegicus | Glutamate receptor ionotropic, kainate 1 |
| P22756 | GRIK1_RAT | Rattus norvegicus | Glutamate receptor ionotropic, kainate 1 |
