PDB Information

PDB5LV2
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors.
Halby, L., Marechal, N., Pechalrieu, D., Cura, V., Franchini, D.M., Faux, C., Alby, F., Troffer-Charlier, N., Kudithipudi, S., Jeltsch, A., Aouadi, W., Decroly, E., Guillemot, J.C., Page, P., Ferroud, C., Bonnefond, L., Guianvarc'h, D., Cavarelli, J., Arimondo, P.B.
Philos.Trans.R.Soc.Lond.B Biol.Sci.
HeaderTransferase
Released2016-09-12
Resolution2.290
CATH Insert Date14 Nov, 2017

PDB Images (25)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped
E 14 Nov, 2017 Chopped
F 14 Nov, 2017 Chopped
G 14 Nov, 2017 Chopped
H 14 Nov, 2017 Chopped

CATH Domains (16)

Domain ID Date inserted into CATH Superfamily CATH Status
5lv2A01 16 Dec, 2017 3.40.50.150 Assigned
5lv2A02 16 Dec, 2017 2.70.160.11 Assigned
5lv2B01 16 Dec, 2017 3.40.50.150 Assigned
5lv2B02 16 Dec, 2017 2.70.160.11 Assigned
5lv2C01 16 Dec, 2017 3.40.50.150 Assigned
5lv2C02 16 Dec, 2017 2.70.160.11 Assigned
5lv2D01 16 Dec, 2017 3.40.50.150 Assigned
5lv2D02 16 Dec, 2017 2.70.160.11 Assigned
5lv2E01 16 Dec, 2017 3.40.50.150 Assigned
5lv2E02 16 Dec, 2017 2.70.160.11 Assigned
5lv2F01 16 Dec, 2017 3.40.50.150 Assigned
5lv2F02 16 Dec, 2017 2.70.160.11 Assigned
5lv2G01 16 Dec, 2017 3.40.50.150 Assigned
5lv2G02 16 Dec, 2017 2.70.160.11 Assigned
5lv2H01 16 Dec, 2017 3.40.50.150 Assigned
5lv2H02 16 Dec, 2017 2.70.160.11 Assigned

UniProtKB Entries (8)

Accession Gene ID Taxon Description
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1
Q9WVG6 CARM1_MOUSE Mus musculus Histone-arginine methyltransferase CARM1