PDB Information

PDB5LOF
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceEscherichia coli O157:H7
Primary Citation
The MCL1 inhibitor S63845 is tolerable and effective in diverse cancer models.
Kotschy, A., Szlavik, Z., Murray, J., Davidson, J., Maragno, A.L., Le Toumelin-Braizat, G., Chanrion, M., Kelly, G.L., Gong, J.N., Moujalled, D.M., Bruno, A., Csekei, M., Paczal, A., Szabo, Z.B., Sipos, S., Radics, G., Proszenyak, A., Balint, B., Ondi, L., Blasko, G., Robertson, A., Surgenor, A., Dokurno, P., Chen, I., Matassova, N., Smith, J., Pedder, C., Graham, C., Studeny, A., Lysiak-Auvity, G., Girard, A.M., Grave, F., Segal, D., Riffkin, C.D., Pomilio, G., Galbraith, L.C., Aubrey, B.J., Brennan, M.S., Herold, M.J., Chang, C., Guasconi, G., Cauquil, N., Melchiore, F., Guigal-Stephan, N., Lockhart, B., Colland, F., Hickman, J.A., Roberts, A.W., Huang, D.C., Wei, A.H., Strasser, A., Lessene, G., Geneste, O.
Nature
HeaderApoptosis/Inhibitor
Released2016-08-09
Resolution2.200
CATH Insert Date06 Nov, 2016

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Nov, 2016 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P0AEY0 MALE_ECO57 Escherichia coli O157:H7 Maltose/maltodextrin-binding periplasmic protein
Q07820 MCL1_HUMAN Homo sapiens Induced myeloid leukemia cell differentiation protein Mcl-1