PDB Information

PDB5L4Q
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Synthesis and Structure-Activity Relationships of 3,5-Disubstituted-pyrrolo[2,3- b]pyridines as Inhibitors of Adaptor-Associated Kinase 1 with Antiviral Activity.
Verdonck, S., Pu, S.Y., Sorrell, F.J., Elkins, J.M., Froeyen, M., Gao, L.J., Prugar, L.I., Dorosky, D.E., Brannan, J.M., Barouch-Bentov, R., Knapp, S., Dye, J.M., Herdewijn, P., Einav, S., De Jonghe, S.
J.Med.Chem.
HeaderTransferase
Released2016-05-26
Resolution1.970
CATH Insert Date19 Jun, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 20 Jun, 2016 Chopped
B 20 Jun, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5l4qA00 20 Jul, 2016 1.10.510.10 Assigned
5l4qB00 21 Jul, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q2M2I8 AAK1_HUMAN Homo sapiens AP2-associated protein kinase 1
Q2M2I8 AAK1_HUMAN Homo sapiens AP2-associated protein kinase 1