PDB Information

PDB5L01
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K-12
Gene SourceHomo sapiens
Primary Citation
Optimization of spirocyclic proline tryptophan hydroxylase-1 inhibitors.
Goldberg, D.R., De Lombaert, S., Aiello, R., Bourassa, P., Barucci, N., Zhang, Q., Paralkar, V., Stein, A.J., Holt, M., Valentine, J., Zavadoski, W.
Bioorg. Med. Chem. Lett.
HeaderOxidoreductase/Inhibitor
Released2016-07-26
Resolution1.900
CATH Insert Date07 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5l01A00 14 Dec, 2017 1.10.800.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P17752 TPH1_HUMAN Homo sapiens Tryptophan 5-hydroxylase 1