PDB Information

PDB5KYK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Covalent Guanosine Mimetic Inhibitors of G12C KRAS.
Xiong, Y., Lu, J., Hunter, J., Li, L., Scott, D., Choi, H.G., Lim, S.M., Manandhar, A., Gondi, S., Sim, T., Westover, K.D., Gray, N.S.
ACS Med Chem Lett
HeaderHydrolase/Hydrolase Inhibitor
Released2016-07-21
Resolution2.700
CATH Insert Date07 May, 2017

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
C 08 May, 2017 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
5kykA00 13 May, 2017 3.40.50.300 Assigned
5kykB00 14 May, 2017 3.40.50.300 Assigned
5kykC00 14 May, 2017 3.40.50.300 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas