PDB 5kyk
PDB Information
PDB | 5KYK |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21(DE3) |
Gene Source | Homo sapiens |
Primary Citation | Covalent Guanosine Mimetic Inhibitors of G12C KRAS.
ACS Med Chem Lett
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2016-07-21 |
Resolution | 2.700 |
CATH Insert Date | 07 May, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (3)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 May, 2017 | Chopped |
B | 08 May, 2017 | Chopped |
C | 08 May, 2017 | Chopped |
CATH Domains (3)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5kykA00 | 13 May, 2017 | 3.40.50.300 | Assigned |
5kykB00 | 14 May, 2017 | 3.40.50.300 | Assigned |
5kykC00 | 14 May, 2017 | 3.40.50.300 | Assigned |
UniProtKB Entries (3)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P01116 | RASK_HUMAN | Homo sapiens | GTPase KRas |
P01116 | RASK_HUMAN | Homo sapiens | GTPase KRas |
P01116 | RASK_HUMAN | Homo sapiens | GTPase KRas |