PDB 5kyj
PDB Information
PDB | 5KYJ |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core.
Bioorg.Med.Chem.Lett.
|
Header | Dna Binding Protein |
Released | 2016-07-21 |
Resolution | 2.800 |
CATH Insert Date | 09 Oct, 2016 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 10 Oct, 2016 | Chopped |
B | 10 Oct, 2016 | Chopped |
E | 10 Oct, 2016 | Chopped |
F | 10 Oct, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5kyjA00 | 30 Nov, 2016 | 1.10.565.10 | Assigned |
5kyjB00 | 03 Jul, 2018 | 1.10.565.10 | Assigned |
5kyjE00 | 30 Nov, 2016 | 1.10.565.10 | Assigned |
5kyjF00 | 03 Jul, 2018 | 1.10.565.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P28702 | RXRB_HUMAN | Homo sapiens | Retinoic acid receptor RXR-beta |
P28702 | RXRB_HUMAN | Homo sapiens | Retinoic acid receptor RXR-beta |
P55055 | NR1H2_HUMAN | Homo sapiens | Oxysterols receptor LXR-beta |
P55055 | NR1H2_HUMAN | Homo sapiens | Oxysterols receptor LXR-beta |