PDB Information

PDB5KTW
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a Potent and Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300.
Crawford, T.D., Romero, F.A., Lai, K.W., Tsui, V., Taylor, A.M., de Leon Boenig, G., Noland, C.L., Murray, J., Ly, J., Choo, E.F., Hunsaker, T.L., Chan, E.W., Merchant, M., Kharbanda, S., Gascoigne, K.E., Kaufman, S., Beresini, M.H., Liao, J., Liu, W., Chen, K.X., Chen, Z., Conery, A.R., Cote, A., Jayaram, H., Jiang, Y., Kiefer, J.R., Kleinheinz, T., Li, Y., Maher, J., Pardo, E., Poy, F., Spillane, K.L., Wang, F., Wang, J., Wei, X., Xu, Z., Xu, Z., Yen, I., Zawadzke, L., Zhu, X., Bellon, S., Cummings, R., Cochran, A.G., Albrecht, B.K., Magnuson, S.
J. Med. Chem.
HeaderTransferase
Released2016-07-12
Resolution1.090
CATH Insert Date20 Nov, 2016

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 21 Nov, 2016 Chopped
B 21 Nov, 2016 Chopped
C 21 Nov, 2016 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
5ktwA00 25 Nov, 2016 1.20.920.10 Assigned
5ktwB00 24 Nov, 2016 1.20.920.10 Assigned
5ktwC00 25 Nov, 2016 1.20.920.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein