PDB Information

PDB5KRS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
A New Class of Allosteric HIV-1 Integrase Inhibitors Identified by Crystallographic Fragment Screening of the Catalytic Core Domain.
Patel, D., Antwi, J., Koneru, P.C., Serrao, E., Forli, S., Kessl, J.J., Feng, L., Deng, N., Levy, R.M., Fuchs, J.R., Olson, A.J., Engelman, A.N., Bauman, J.D., Kvaratskhelia, M., Arnold, E.
J.Biol.Chem.
HeaderHydrolase, Transferase/Inhibitor
Released2016-07-07
Resolution1.700
CATH Insert Date09 Oct, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5krsA00 15 Oct, 2016 3.30.420.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q76353 Q76353_9HIV1 Human immunodeficiency virus 1 Integrase