PDB 5kr7

PDB Information

PDB5KR7
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification of potent, selective KDM5 inhibitors.
Gehling, V.S., Bellon, S.F., Harmange, J.C., LeBlanc, Y., Poy, F., Odate, S., Buker, S., Lan, F., Arora, S., Williamson, K.E., Sandy, P., Cummings, R.T., Bailey, C.M., Bergeron, L., Mao, W., Gustafson, A., Liu, Y., VanderPorten, E., Audia, J.E., Trojer, P., Albrecht, B.K.
Bioorg.Med.Chem.Lett.
HeaderOxidoreductase
Released2016-07-07
Resolution1.900
CATH Insert Date04 Sep, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Sep, 2016 Chopped
B 05 Sep, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5kr7A01 09 Sep, 2016 2.60.120.650 Assigned
5kr7B01 08 Sep, 2016 2.60.120.650 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H3R0 KDM4C_HUMAN Homo sapiens Lysine-specific demethylase 4C
Q9H3R0 KDM4C_HUMAN Homo sapiens Lysine-specific demethylase 4C