PDB Information

PDB5KJK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design, Synthesis, and Biological Activity of Substrate Competitive SMYD2 Inhibitors.
Cowen, S.D., Russell, D., Dakin, L.A., Chen, H., Larsen, N.A., Godin, R., Throner, S., Zheng, X., Molina, A., Wu, J., Cheung, T., Howard, T., Garcia-Arenas, R., Keen, N., Pendleton, C.S., Pietenpol, J.A., Ferguson, A.D.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2016-06-20
Resolution1.930
CATH Insert Date25 Dec, 2016

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 26 Dec, 2016 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
5kjkA01 30 Dec, 2016 2.170.270.10 Assigned
5kjkA02 30 Dec, 2016 Holding pen
5kjkA03 30 Dec, 2016 1.25.40.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9NRG4 SMYD2_HUMAN Homo sapiens N-lysine methyltransferase SMYD2