PDB Information

PDB5KCX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors - Part I.
Barberis, C., Moorcroft, N., Arendt, C., Levit, M., Moreno-Mazza, S., Batchelor, J., Mechin, I., Majid, T.
Bioorg. Med. Chem. Lett.
HeaderTransferase/Inhibitor
Released2016-06-07
Resolution2.200
CATH Insert Date14 Nov, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5kcxA01 10 Dec, 2017 3.30.200.20 Assigned
5kcxA02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1