PDB 5kby
PDB Information
| PDB | 5KBY | 
| Method | X-RAY DIFFRACTION | 
| Host Organism | unidentified baculovirus | 
| Gene Source | Homo sapiens | 
| Primary Citation | Trelagliptin (SYR-472, Zafatek), Novel Once-Weekly Treatment for Type 2 Diabetes, Inhibits Dipeptidyl Peptidase-4 (DPP-4) via a Non-Covalent Mechanism. Plos One | 
| Header | Hydrolase/Hydrolase Inhibitor | 
| Released | 2016-06-03 | 
| Resolution | 2.240 | 
| CATH Insert Date | 24 Jul, 2016 | 
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status | 
|---|---|---|
| A | 25 Jul, 2016 | Chopped | 
| B | 25 Jul, 2016 | Chopped | 
| C | 25 Jul, 2016 | Chopped | 
| D | 25 Jul, 2016 | Chopped | 
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status | 
|---|---|---|---|
| 5kbyA01 | 01 Sep, 2016 | 2.140.10.30 | Assigned | 
| 5kbyA02 | 01 Sep, 2016 | 3.40.50.1820 | Assigned | 
| 5kbyB01 | 01 Sep, 2016 | 2.140.10.30 | Assigned | 
| 5kbyB02 | 01 Sep, 2016 | 3.40.50.1820 | Assigned | 
| 5kbyC01 | 01 Sep, 2016 | 2.140.10.30 | Assigned | 
| 5kbyC02 | 01 Sep, 2016 | 3.40.50.1820 | Assigned | 
| 5kbyD01 | 01 Sep, 2016 | 2.140.10.30 | Assigned | 
| 5kbyD02 | 01 Sep, 2016 | 3.40.50.1820 | Assigned | 
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description | 
|---|---|---|---|
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 | 
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 | 
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 | 
| P27487 | DPP4_HUMAN | Homo sapiens | Dipeptidyl peptidase 4 | 
