PDB 5kbq
PDB Information
| PDB | 5KBQ |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
ACS Med Chem Lett
|
| Header | Transferase |
| Released | 2016-06-03 |
| Resolution | 2.580 |
| CATH Insert Date | 09 Oct, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 10 Oct, 2016 | Chopped |
| B | 10 Oct, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5kbqA01 | 15 Oct, 2016 | 3.30.200.20 | Assigned |
| 5kbqA02 | 15 Oct, 2016 | 1.10.510.10 | Assigned |
| 5kbqB01 | 15 Oct, 2016 | 3.30.200.20 | Assigned |
| 5kbqB02 | 15 Oct, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |
| Q13153 | PAK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase PAK 1 |
