PDB Information

PDB5KAO
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
A Modified P1 Moiety Enhances In Vitro Antiviral Activity against Various Multidrug-Resistant HIV-1 Variants and In Vitro Central Nervous System Penetration Properties of a Novel Nonpeptidic Protease Inhibitor, GRL-10413.
Amano, M., Salcedo-Gomez, P.M., Zhao, R., Yedidi, R.S., Das, D., Bulut, H., Delino, N.S., Sheri, V.R., Ghosh, A.K., Mitsuya, H.
Antimicrob.Agents Chemother.
HeaderHydrolase/Hydrolase Inhibitor
Released2016-06-01
Resolution1.800
CATH Insert Date16 Oct, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Oct, 2016 Chopped
B 17 Oct, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5kaoA00 22 Oct, 2016 2.40.70.10 Assigned
5kaoB00 21 Oct, 2016 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein
P04585 POL_HV1H2 HIV-1 M:B_HXB2R Gag-Pol polyprotein