PDB 5k0x
PDB Information
PDB | 5K0X |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Discovery of Macrocyclic Pyrimidines as MerTK-Specific Inhibitors.
ChemMedChem
|
Header | Transferase/Transferase Inhibitor |
Released | 2016-05-17 |
Resolution | 2.230 |
CATH Insert Date | 07 May, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 May, 2017 | Chopped |
B | 08 May, 2017 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5k0xA01 | 13 May, 2017 | Holding pen | |
5k0xA02 | 13 May, 2017 | 1.10.510.10 | Assigned |
5k0xB01 | 13 May, 2017 | Holding pen | |
5k0xB02 | 13 May, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer |
Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer |