PDB Information

PDB5K0X
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Macrocyclic Pyrimidines as MerTK-Specific Inhibitors.
McIver, A.L., Zhang, W., Liu, Q., Jiang, X., Stashko, M.A., Nichols, J., Miley, M.J., Norris-Drouin, J., Machius, M., DeRyckere, D., Wood, E., Graham, D.K., Earp, H.S., Kireev, D., Frye, S.V., Wang, X.
ChemMedChem
HeaderTransferase/Transferase Inhibitor
Released2016-05-17
Resolution2.230
CATH Insert Date07 May, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5k0xA01 13 May, 2017 Holding pen
5k0xA02 13 May, 2017 1.10.510.10 Assigned
5k0xB01 13 May, 2017 Holding pen
5k0xB02 13 May, 2017 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q12866 MERTK_HUMAN Homo sapiens Tyrosine-protein kinase Mer
Q12866 MERTK_HUMAN Homo sapiens Tyrosine-protein kinase Mer