PDB Information

PDB5K03
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceRattus norvegicus
Primary Citation
Design of Potent and Druglike Nonphenolic Inhibitors for Catechol O-Methyltransferase Derived from a Fragment Screening Approach Targeting the S-Adenosyl-l-methionine Pocket.
Lerner, C., Jakob-Roetne, R., Buettelmann, B., Ehler, A., Rudolph, M., Rodriguez Sarmiento, R.M.
J. Med. Chem.
HeaderTransferase
Released2016-05-17
Resolution1.810
CATH Insert Date02 Oct, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 03 Oct, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5k03A00 20 Oct, 2016 3.40.50.150 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P22734 COMT_RAT Rattus norvegicus Catechol O-methyltransferase