PDB Information

PDB5JZS
MethodX-RAY DIFFRACTION
Host OrganismPseudomonas putida
Gene SourceMycobacterium tuberculosis
Primary Citation
Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach.
Ryan, A., Polycarpou, E., Lack, N.A., Evangelopoulos, D., Sieg, C., Halman, A., Bhakta, S., Eleftheriadou, O., McHugh, T.D., Keany, S., Lowe, E.D., Ballet, R., Abuhammad, A., Jacobs, W.R., Ciulli, A., Sim, E.
Br. J. Pharmacol.
HeaderHydrolase
Released2016-05-17
Resolution2.270
CATH Insert Date07 May, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5jzsA00 13 May, 2017 3.40.50.1820 Assigned
5jzsB00 13 May, 2017 3.40.50.1820 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P9WNH5 HSAD_MYCTU Mycobacterium tuberculosis H37Rv 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase
P9WNH5 HSAD_MYCTU Mycobacterium tuberculosis H37Rv 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase