PDB Information

PDB5JAN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening.
Woolford, A.J., Pero, J.E., Aravapalli, S., Berdini, V., Coyle, J.E., Day, P.J., Dodson, A.M., Grondin, P., Holding, F.P., Lee, L.Y., Li, P., Manas, E.S., Marino, J., Martin, A.C., McCleland, B.W., McMenamin, R.L., Murray, C.W., Neipp, C.E., Page, L.W., Patel, V.K., Potvain, F., Rich, S., Rivero, R.A., Smith, K., Somers, D.O., Trottet, L., Velagaleti, R., Williams, G., Xie, R.
J.Med.Chem.
HeaderHydrolase
Released2016-04-12
Resolution2.120
CATH Insert Date05 Jun, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 06 Jun, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5janA00 19 Jul, 2016 3.40.50.1820 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q13093 PAFA_HUMAN Homo sapiens Platelet-activating factor acetylhydrolase