PDB 5j1v
PDB Information
| PDB | 5J1V |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.
Eur.J.Med.Chem.
|
| Header | Transferase |
| Released | 2016-03-29 |
| Resolution | 2.520 |
| CATH Insert Date | 15 May, 2016 |
PDB Images (9)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 May, 2016 | Chopped |
| B | 16 May, 2016 | Chopped |
| C | 16 May, 2016 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5j1vA01 | 30 Nov, 2016 | 3.30.200.20 | Assigned |
| 5j1vA02 | 30 Nov, 2016 | 1.10.510.10 | Assigned |
| 5j1vB01 | 30 Nov, 2016 | 3.30.200.20 | Assigned |
| 5j1vB02 | 30 Nov, 2016 | 1.10.510.10 | Assigned |
| 5j1vC00 | 29 Nov, 2016 | Holding pen |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P49759 | CLK1_HUMAN | Homo sapiens | Dual specificity protein kinase CLK1 |
| P49759 | CLK1_HUMAN | Homo sapiens | Dual specificity protein kinase CLK1 |
| P49759 | CLK1_HUMAN | Homo sapiens | Dual specificity protein kinase CLK1 |
