PDB 5itd
PDB Information
| PDB | 5ITD |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors.
Acs Med.Chem.Lett.
|
| Header | Transferase/Protein Transport/Inhibitor |
| Released | 2016-03-16 |
| Resolution | 3.020 |
| CATH Insert Date | 09 Oct, 2016 |
PDB Images (10)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 10 Oct, 2016 | Chopped |
| B | 10 Oct, 2016 | Chopped |
CATH Domains (7)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5itdA01 | 12 Jul, 2018 | Check for files | |
| 5itdA02 | 12 Jul, 2018 | Check for files | |
| 5itdA03 | 12 Jul, 2018 | Check for files | |
| 5itdA04 | 12 Jul, 2018 | Check for files | |
| 5itdA05 | 12 Jul, 2018 | Check for files | |
| 5itdB01 | 14 Nov, 2017 | Holding pen | |
| 5itdB02 | 14 Nov, 2017 | 1.10.287.1490 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P27986 | P85A_HUMAN | Homo sapiens | Phosphatidylinositol 3-kinase regulatory subunit alpha |
| P42336 | PK3CA_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
