PDB Information

PDB5I8A
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Potent, selective and orally bioavailable leucine-rich repeat kinase 2 (LRRK2) inhibitors.
Greshock, T.J., Sanders, J.M., Drolet, R.E., Rajapakse, H.A., Chang, R.K., Kim, B., Rada, V.L., Tiscia, H.E., Su, H., Lai, M.T., Sur, S.M., Sanchez, R.I., Bilodeau, M.T., Renger, J.J., Kern, J.T., McCauley, J.A.
Bioorg. Med. Chem. Lett.
HeaderTransferase/Transferase Inhibitor
Released2016-02-18
Resolution2.330
CATH Insert Date14 Nov, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5i8aA01 10 Dec, 2017 3.30.200.20 Assigned
5i8aA02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P04629 NTRK1_HUMAN Homo sapiens High affinity nerve growth factor receptor