PDB Information

PDB5HRX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis.
Myrianthopoulos, V., Gaboriaud-Kolar, N., Tallant, C., Hall, M.L., Grigoriou, S., Brownlee, P.M., Fedorov, O., Rogers, C., Heidenreich, D., Wanior, M., Drosos, N., Mexia, N., Savitsky, P., Bagratuni, T., Kastritis, E., Terpos, E., Filippakopoulos, P., Muller, S., Skaltsounis, A.L., Downs, J.A., Knapp, S., Mikros, E.
J.Med.Chem.
HeaderTranscription
Released2016-01-24
Resolution1.730
CATH Insert Date06 Nov, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Nov, 2016 Chopped
B 07 Nov, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5hrxA00 09 Nov, 2016 1.20.920.10 Assigned
5hrxB00 10 Nov, 2016 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1
Q86U86 PB1_HUMAN Homo sapiens Protein polybromo-1