PDB Information

PDB5HO7
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of novel 7-azaindoles as PDK1 inhibitors.
Wucherer-Plietker, M., Merkul, E., Muller, T.J., Esdar, C., Knochel, T., Heinrich, T., Buchstaller, H.P., Greiner, H., Dorsch, D., Finsinger, D., Calderini, M., Bruge, D., Gradler, U.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2016-01-19
Resolution3.000
CATH Insert Date19 Jun, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Jun, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ho7A01 17 Jul, 2016 3.30.200.20 Assigned
5ho7A02 17 Jul, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1