PDB Information

PDB5H8B
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo.
Dowling, J.E., Alimzhanov, M., Bao, L., Chuaqui, C., Denz, C.R., Jenkins, E., Larsen, N.A., Lyne, P.D., Pontz, T., Ye, Q., Holdgate, G.A., Snow, L., O'Connell, N., Ferguson, A.D.
Acs Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2015-12-23
Resolution2.550
CATH Insert Date10 Apr, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5h8bA01 13 May, 2016 1.10.510.10 Assigned
5h8bA02 13 May, 2016 3.30.200.20 Assigned
5h8bB01 13 May, 2016 1.10.510.10 Assigned
5h8bB02 13 May, 2016 3.30.200.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha