PDB Information

PDB5H1U
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli 'BL21-Gold(DE3)pLysS AG'
Gene SourceHomo sapiens
Primary Citation
The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network
Liu, J., Li, F., Bao, H., Jiang, Y., Zhang, S., Ma, R., Gao, J., Wu, J., Ruan, K.
FEBS J.
HeaderTranscription/Transcription Inhibitor
Released2016-10-11
Resolution1.900
CATH Insert Date07 May, 2017

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
C 08 May, 2017 Chopped
D 08 May, 2017 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5h1uA01 12 May, 2017 3.30.40.10 Assigned
5h1uA02 12 May, 2017 1.20.920.10 Assigned
5h1uB01 12 May, 2017 3.30.40.10 Assigned
5h1uB02 12 May, 2017 1.20.920.10 Assigned
5h1uC01 12 May, 2017 3.30.40.10 Assigned
5h1uC02 12 May, 2017 1.20.920.10 Assigned
5h1uD01 12 May, 2017 3.30.40.10 Assigned
5h1uD02 12 May, 2017 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O15164 TIF1A_HUMAN Homo sapiens Transcription intermediary factor 1-alpha
O15164 TIF1A_HUMAN Homo sapiens Transcription intermediary factor 1-alpha
O15164 TIF1A_HUMAN Homo sapiens Transcription intermediary factor 1-alpha
O15164 TIF1A_HUMAN Homo sapiens Transcription intermediary factor 1-alpha