PDB 5h1u
PDB Information
| PDB | 5H1U |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli 'BL21-Gold(DE3)pLysS AG' |
| Gene Source | Homo sapiens |
| Primary Citation | The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network
FEBS J.
|
| Header | Transcription/Transcription Inhibitor |
| Released | 2016-10-11 |
| Resolution | 1.900 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
| C | 08 May, 2017 | Chopped |
| D | 08 May, 2017 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5h1uA01 | 12 May, 2017 | 3.30.40.10 | Assigned |
| 5h1uA02 | 12 May, 2017 | 1.20.920.10 | Assigned |
| 5h1uB01 | 12 May, 2017 | 3.30.40.10 | Assigned |
| 5h1uB02 | 12 May, 2017 | 1.20.920.10 | Assigned |
| 5h1uC01 | 12 May, 2017 | 3.30.40.10 | Assigned |
| 5h1uC02 | 12 May, 2017 | 1.20.920.10 | Assigned |
| 5h1uD01 | 12 May, 2017 | 3.30.40.10 | Assigned |
| 5h1uD02 | 12 May, 2017 | 1.20.920.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O15164 | TIF1A_HUMAN | Homo sapiens | Transcription intermediary factor 1-alpha |
| O15164 | TIF1A_HUMAN | Homo sapiens | Transcription intermediary factor 1-alpha |
| O15164 | TIF1A_HUMAN | Homo sapiens | Transcription intermediary factor 1-alpha |
| O15164 | TIF1A_HUMAN | Homo sapiens | Transcription intermediary factor 1-alpha |
