PDB Information

PDB5G3M
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Azd2716: A Novel Secreted Phospholipase A2 (Spla2) Inhibitor for the Treatment of Coronary Artery Disease
Giordanetto, F., Pettersen, D., Starke, I., Nordberg, P., Dahlstrom, M., Knerr, L., Selmi, N., Rosengren, B., Larsson, L.O., Sandmark, J., Castaldo, M., Dekker, N., Karlsson, U., Hurt-Camejo, E.
Acs Med.Chem.Lett.
HeaderHydrolase
Released2016-04-29
Resolution1.850
CATH Insert Date02 Oct, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Oct, 2016 Chopped
B 03 Oct, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5g3mA00 07 Oct, 2016 1.20.90.10 Assigned
5g3mB00 07 Oct, 2016 1.20.90.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2