PDB Information

PDB5G2N
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Discovery and Sar of Novel 2,3-Dihydroimidazo(1,2-C)Quinazoline Pi3K Inhibitors: Identification of Copanlisib (Bay 80-6946)
Schaefer, M., Scott, W.J., Hentemann, M.F., Rowley, R.B., Bull, C.O., Jenkins, S., Bullion, A.M., Johnson, J., Redman, A., Robbins, A.H., Esler, W., Fracasso, R.P., Garrison, T., Hamilton, M., Michels, M., Wood, J.E., Wilkie, D.P., Xiao, H., Levy, J., Liu, N., Stasik, E., Brands, M., Lefranc, J.
Chemmedchem
HeaderTransferase
Released2016-04-11
Resolution2.680
CATH Insert Date24 Apr, 2016

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 25 Apr, 2016 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5g2nA01 12 May, 2016 3.10.20.90 Assigned
5g2nA02 12 May, 2016 2.60.40.150 Assigned
5g2nA03 12 May, 2016 1.25.40.70 Assigned
5g2nA04 12 May, 2016 3.30.1010.10 Assigned
5g2nA05 12 May, 2016 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform